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Chemicals
[D-Ala2] Deltorphin I CAS NO.122752-15-2
<p>[D-Ala2] Deltorphin I is a synthetic heptapeptide analog derived from frog skin secretion, engineered with a D-amino acid substitution to enhance its metabolic stability and receptor selectivity. It functions as a highly potent and selective agonist for the delta-opioid receptor (DOR), making it a critical tool in neuropharmacology research for studying pain pathways and receptor signaling without the rapid degra…
SupplierGlobal Technology Co., Ltd.www.hqtechtirz.com
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About this product
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TECHNICAL SPECIFICATIONS
| Item | Specification |
|---|---|
| Product Name | [D-Ala2] Deltorphin I |
| CAS NO. | 122752-15-2 |
| Appearance | White to off-white lyophilized powder |
| Molecular Formula | C₃₇H₅₂N₈O₁₀ |
| Molecular Weight | 768.9g/mol |
| Purity (RP-HPLC) | ≥95% |
| Solubility | Soluble in water, dilute acetic acid, or DMSO |
| Endotoxin | ≤1 EU/mg |
| Biological Activity | Potent and selective agonist for the delta-opioid receptor (DOR) |
| Storage Conditions | Store at -20°C, protected from moisture and light |
| Stock Location | Stock in USA |
| MOQ | 1g |
1.MECHANISM OF ACTION
The peptide exerts its effects by binding with high affinity specifically to the delta-opioid receptor (DOR) in the central nervous system. Upon binding, it activates G-protein coupled signaling pathways, leading to the inhibition of adenylate cyclase and a reduction in intracellular cAMP levels. This action modulates neuronal excitability and neurotransmitter release, effectively producing potent analgesic and antinociceptive effects in experimental models.
2.PRODUCT INDICATIONS
This product is indicated for preclinical research applications, primarily in the fields of neuroscience and pharmacology. It is used to investigate DOR-mediated analgesia, study the mechanisms of opioid tolerance and dependence, and screen for novel analgesic drugs. Researchers also utilize it in receptor binding assays and animal models of chronic pain to elucidate the role of delta receptors in stress and emotional behavior.
3.CLINICAL EFFICACY OF PRODUCT
In experimental studies, [D-Ala2] Deltorphin I has demonstrated significant efficacy in producing antinociception and reducing pain responses in rodent models. It shows a high potency at the receptor level, though chronic administration studies reveal the development of tolerance, which is a key area of investigation for understanding opioid-related side effects. Its research-grade performance supports drug discovery efforts aimed at developing non-addictive pain therapies.
4.Certificate
GlobalTech Co., Ltd. is committed to providing high-purity biotechnological peptide products, adhering strictly to quality standards and obtaining internationally recognized certifications.
Our production partners all employ GMP-compliant production systems and possess standardized quality control processes covering raw material procurement, synthesis, purification, testing, packaging, and storage. Each batch of product comes with complete documentation, including a Certificate of Analysis (COA), HPLC purity report, mass spectrometry (MS) chromatograms, and third-party testing reports available upon request.
We prioritize:
1.A rigorous quality management system
2.Batch traceability and stability data
3.Professional laboratory testing and validation
4.Compliance with international trade standards
Our commitment to quality, transparency, and regulatory compliance ensures the provision of reliable, stable, and research-grade peptide products to our global partners.
5.DELIVERY & SHIPPING
We specialize in global logistics for various cosmetic peptides. Your order will be handled with the utmost care, ensuring safe, reliable, and intact delivery.
Professional and Secure Packaging
Each bottle of peptide is protected with a special packaging solution to ensure stability and integrity during transportation.
We can also customize packaging according to customer needs.
Shipping Methods
Main Method: International Air Freight
We primarily use DHL, FedEx, UPS, and TNT because of their global reliability, speed, and advanced tracking systems. Air freight ensures the fastest transit time and minimizes the impact of environmental factors on the product.
Global Technology Co., Ltd. is a modern and advanced enterprise specializing in the production and export of active pharmaceutical ingredients (APIs), peptides, and plant extracts. The company invests in and collaborates closely with domestic manufacturers holding GMP, DMF, and FDA certifications, as well as laboratories at renowned universities, to meet diverse customer needs ranging from gram-level to ton-level. This enables Dejurui Pharmaceutical to provide customers with more flexible and convenient access to cost-effective, high-quality products and superior services.
We focus on the research and development and supply of high-quality chemical products, strictly adhering to international standards and quality systems. Our products are stable in performance and reliable in purity, widely used in industrial manufacturing, scientific research, and the fine chemical industry. We provide solid support at every stage with a professional and responsible attitude.
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